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BCR-ABL

7 drugs

BCR-ABL1 Fusion Gene (Philadelphia Chromosome)

Predictive biomarker for patient selection in 3 indications

Understanding BCR-ABL

What it means: BCR-ABL results from a translocation creating the Philadelphia chromosome. The fusion protein has constitutive tyrosine kinase activity.
Why it matters: Tyrosine kinase inhibitors (imatinib, dasatinib, nilotinib, ponatinib) revolutionized CML treatment, achieving long-term remissions.
Testing: Tested via cytogenetics, FISH, or RT-PCR. Quantitative PCR monitors treatment response (molecular response levels).
7
Approved Drugs
3
Indications
6
Companies

BCR-ABL is a precision-medicine biomarker linked to 7 FDA-approved targeted drugs from 6 companies, spanning 3 indications including Chronic Myeloid Leukemia, Acute Lymphoblastic Leukemia, Chronic Myelogenous Leukemia. Explore the targeted therapies, indications, testing methods, and companies developing BCR-ABL drugs below.

Search BCR-ABL Clinical Trials

Search recruiting trials on ClinicalTrials.gov

Drugs Targeting BCR-ABL

Drug Company Therapeutic Area
BOSULIF PF PRISM CV Oncology
DANZITEN AZURITY Oncology
DASATINIB Apotex Oncology
PHYRAGO HANDA THERAP Oncology
SCEMBLIX Novartis Oncology
SPRYCEL Bristol-Myers Squibb Oncology
TASIGNA Novartis Oncology

BCR-ABL Indications

Chronic Myeloid Leukemia Acute Lymphoblastic Leukemia Chronic Myelogenous Leukemia