TheraRadar
Dashboards /MOA Platforms
Data updated: Jun 28, 2026

MOA Platform Heatmaps

Pick a mechanism-of-action family and see every drug against that target across all indications — “all assets against target X.” Each grid is drugs (rows) × indications (columns), with forward catalysts and per-asset detail.

19 curated families · 632 drugs mapped

IO checkpoint inhibitors

Pro

PD-1, PD-L1, CTLA-4, LAG-3, TIGIT, TIM-3 antibodies and bispecifics — the most-mature IO landscape.

116 drugs 37 indications 510 trials 64 Ph3

Antibody-drug conjugates (ADCs)

Pro

Antibody-drug conjugates spanning multiple tumor antigens. The dominant emerging modality across solid tumors.

52 drugs 33 indications 366 trials 27 Ph3

T-cell engagers (CD3 bispecifics)

Pro

Bispecific antibodies engaging T-cells via CD3 to a tumor antigen. The fastest-growing class in oncology after IO and ADCs.

39 drugs 32 indications 208 trials 20 Ph3

GLP-1 / incretin agonists

Pro

GLP-1 and multi-incretin (GIP, glucagon, amylin) agonists across obesity, type 2 diabetes, MASH, and cardiometabolic — the highest-value cross-indication race in pharma.

35 drugs 25 indications 204 trials 23 Ph3

EGFR family inhibitors

Pro

EGFR TKIs across generations, exon-20 selective, bispecifics, and EGFR ADCs.

56 drugs 24 indications 201 trials 21 Ph3

CD19-targeted therapies

Pro

CD19-directed therapies across modalities (CAR-T, T-cell-engaging bispecifics, mAb/ADC) AND across domains — the heme-oncology workhorse (lymphoma/leukemia) now crossing into autoimmune disease (lupus, myasthenia, scleroderma, myositis), where CD19 CAR-T "resets" the B-cell compartment.

70 drugs 30 indications 188 trials 14 Ph3

HER2 family

Pro

HER2 mAbs, ADCs, bispecifics, and small-molecule TKIs.

51 drugs 15 indications 171 trials 22 Ph3

KRAS family inhibitors

Pro

KRAS inhibitors spanning G12C, G12D, G12V, pan-RAS, RAS(ON), KRAS vaccines, and KRAS-targeted TCR-T.

50 drugs 8 indications 125 trials 15 Ph3

JAK / TYK2 inhibitors

Pro

JAK pan / JAK1 / JAK1/2 / JAK3 / TYK2 inhibitors — the oral kinase backbone across immunology, dermatology, myeloproliferative neoplasms, and (emerging) CNS.

21 drugs 29 indications 124 trials 19 Ph3

BCMA-targeted therapies

Pro

BCMA-directed therapies across modalities — CAR-T, T-cell-engaging bispecifics, and ADCs — the dominant target in relapsed/refractory multiple myeloma.

21 drugs 11 indications 100 trials 13 Ph3

CAR-T cell therapy

Pro

Autologous and allogeneic CAR-T cells across hematologic and solid tumor targets.

29 drugs 24 indications 77 trials 7 Ph3

Radioligand therapies

Pro

PSMA / SSTR2 / FAP-targeted radioligand therapies — the fast-emerging precision-oncology modality.

33 drugs 16 indications 63 trials 8 Ph3

PARP / DDR inhibitors

Pro

PARP inhibitors and broader DNA-damage-response (ATR, WEE1) inhibitors.

16 drugs 10 indications 61 trials 8 Ph3

IL-23 axis inhibitors

Pro

IL-12/23 (p40) and IL-23 (p19) inhibitors — the dominant immunology class for psoriasis, IBD, and emerging.

9 drugs 5 indications 58 trials 7 Ph3

TL1A inhibitors

Pro

TL1A antibodies for IBD — the most-crowded emerging mechanism in UC and CD across 6 sponsors.

8 drugs 8 indications 37 trials 3 Ph3

Claudin 18.2 targeting

Pro

Claudin 18.2 mAbs, ADCs, bispecifics, and CAR-T across gastric and PDAC.

11 drugs 7 indications 29 trials 5 Ph3

MTAP synthetic-lethal inhibitors

Pro

PRMT5 and MAT2A inhibitors exploiting MTAP-deletion vulnerability — selective oncology synthetic-lethal class.

6 drugs 6 indications 18 trials 1 Ph3

S1P modulators

Pro

Sphingosine-1-phosphate receptor modulators for UC, MS, and other indications.

6 drugs 5 indications 17 trials 6 Ph3

mRNA neoantigen vaccines

Pro

mRNA-encoded personalized neoantigen and shared antigen cancer vaccines.

3 drugs 7 indications 15 trials 2 Ph3

Data: ClinicalTrials.gov · Curated target-family rosters · Updated weekly.