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Data updated: Jun 28, 2026

LO LOESTRIN FE (ethinyl estradiol) · APIL

Women's Health Approved 2010-10-21

Lo Loestrin Fe is a combination hormonal medication used by women to prevent pregnancy. It combines a progestin called norethindrone acetate with an estrogen called ethinyl estradiol to provide contraceptive protection. This medication helps women manage their reproductive health, though its effectiveness has not been evaluated in patients with a body mass index greater than 35.

How LO LOESTRIN FE Works

This medication works primarily by suppressing ovulation. By using a combination of hormones to prevent the release of an egg from the ovaries, the drug effectively stops pregnancy from occurring.

1
Indication
--
Phase 3 Trials
15
Years on Market

Details

Status
Prescription
First Approved
2010-10-21
Patent Cliff
2029

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Routes
ORAL
Dosage Forms
TABLET

Companies

LO LOESTRIN FE Approval History

2011
2012
2013
2014
2015
2016
2017
2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
7 FDA actions from 2010 to 2022
Apr 2022 SUPPL
Label · Labeling
Oct 2021 SUPPL
Label · Labeling
Oct 2017 SUPPL
Label · Labeling

What LO LOESTRIN FE Treats

1 indications

LO LOESTRIN FE is approved for 1 conditions since its original approval in 2010. These indications span multiple therapeutic areas including oncology, immunology, and more.

Source: FDA Label

LO LOESTRIN FE Boxed Warning

CIGARETTE SMOKING AND SERIOUS CARDIOVASCULAR EVENTS Cigarette smoking increases the risk of serious cardiovascular events from combination oral contraceptive (COC ) use. This risk increases with age , particularly in women over 35 years of age , and with the number of cigarettes smoked . For this reason, COCs should not be used by w omen who are over 35 years of age and smoke [ see Contraindications (4) ] . WARNING : CIGARETTE SMOKING AND SERIOUS CARDIOVASCULAR EVENTS See Full Prescribing Inform...

LO LOESTRIN FE Competitive Set

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Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

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Clinical Trial Registry

2 trials
Trial Sponsor ID Phase Status Title
NCT07340190 CDAK539A12102 2025-521000-22-00 Ph 1 recruiting A Drug-drug Interaction Study to Evaluate the Effects of Pelabresib on the Pharmacokinetics of Repaglinide, Midazolam, and Combined Oral Contraceptive in Patients With Advanced Malignancies
NCT06039826 18533 J1I-MC-GZBV Ph 1 completed A Study of LY3437943 in Postmenopausal Female Participants Who Are Overweight or Obese
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Key Completed Trials

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

LO LOESTRIN FE FDA Label Details

Indications & Usage

FDA Label (PDF)

Lo Loestrin ® Fe is indicated for use by women to prevent pregnancy [ see Clinical Studies ] . The efficacy of Lo Loestrin Fe in women with a body mass index (BMI) of > 35 kg/m 2 has not been evaluated. Lo Loestrin Fe is a combination of norethindrone acetate, a progestin, and ethinyl estradiol, an estrogen, indicated for use by women to prevent pregnancy The efficacy of Lo Loestrin Fe in women with a body mass index of > 35 kg/m 2 has not been evaluated

⚠️ BOXED WARNING

WARNING: CIGARETTE SMOKING AND SERIOUS CARDIOVASCULAR EVENTS Cigarette smoking increases the risk of serious cardiovascular events from combination oral contraceptive (COC ) use. This risk increases with age , particularly in women over 35 years of age , and with the number of cigarettes smoked . Fo...

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1 OB patents · 1 families · 14 international docs across 8 countries

LO LOESTRIN FE Patents & Exclusivity

Latest Patent: Feb 2029

Patents (1 active)

US7704984 Expires Feb 2, 2029
Source: FDA Orange Book

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Patent Timeline

  • Cliff: 2029
  • 1 active patents

Trial Analysis

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Competitive Landscape

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.