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Data updated: Jun 28, 2026

VALTREX (valacyclovir hydrochloride) · GSK

Infectious Disease Approved 1995-06-23

Valtrex is an antiviral medication indicated for the treatment of cold sores (herpes labialis) in adults and pediatric patients (12 years and older) and chickenpox in pediatric patients (2 to <18 years). In adult patients, it is used to treat herpes zoster (shingles) and to manage genital herpes by treating initial or recurrent episodes, providing chronic suppressive therapy, and reducing the risk of transmission. Its efficacy and safety have not been established in immunocompromised patients, except for the suppression of genital herpes in HIV-1-infected adults.

How VALTREX Works

Valacyclovir is a deoxynucleoside analogue DNA polymerase inhibitor. As a prodrug, it is rapidly converted to acyclovir, which selectively inhibits viral DNA polymerase. This action interferes with the DNA replication of $\alpha$-herpes viruses (such as HSV and VZV), thereby preventing viral proliferation.

NDA
Small Molecule
9
Indications
--
Phase 3 Trials
3
Priority Reviews
31
Years on Market

Details

Status
Prescription
First Approved
1995-06-23
Routes
ORAL, Oral
Dosage Forms
TABLET, Tablet

Companies

Active Ingredient: VALACYCLOVIR HYDROCHLORIDE

VALTREX Approval History

1996
1997
1998
1999
2000
2001
2002
2003
2004
2005
2006
2007
2008
2009
2010
2011
2012
2013
2014
2015
2016
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2018
2019
2020
2021
2022
2023
2024
2025
2026
Original
New Indication
New Form
Label Update
66 FDA actions from 1995 to 2025 · 6 indication expansions
Nov 2025 SUPPL
Label · Labeling
Jun 2021 SUPPL
Label · Labeling
Dec 2019 SUPPL
Label · Labeling

What VALTREX Treats

4 indications

VALTREX is approved for 4 conditions since its original approval in 1995. These indications span multiple therapeutic areas including oncology, immunology, and more.

  • Cold Sores
  • Genital Herpes
  • Herpes Zoster
  • Chickenpox
Source: FDA Label

VALTREX Competitive Set

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Three rings of competition based on shared molecular targets and treated indications.

Indication competitors

2

Same indication, different mechanism — what else might this patient receive?

Filters applied: drops same-active-ingredient (505(b)(2) reformulations), route-mismatch (topical vs systemic), and cross-therapeutic-area matches in same-indication rings.

Drugs Similar to VALTREX

FDA-approved drugs for similar conditions. Compare mechanisms and indications to understand treatment alternatives.

ACYCLOVIR
ACYCLOVIR
3 shared
XIROMED
Shared indications:
Herpes ZosterGenital HerpesChickenpox
FAMCICLOVIR
FAMCICLOVIR
2 shared
NATCO PHARMA
Shared indications:
Genital HerpesHerpes Zoster
VALACYCLOVIR HYDROCHLORIDE
VALACYCLOVIR HYDROCHLORIDE
2 shared
AIPING PHARM INC
Shared indications:
Genital herpesChickenpox
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Active Pipeline

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Key Completed Trials

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Completed studies with published results, ranked by significance

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Trial Timeline

Full development history with FDA approval milestones

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Understanding FDA Approval Types
Count Type What it means
- ORIG Original approval - drug first enters market
- SUPPL - Efficacy New indication (new disease/condition approved)
- SUPPL - Labeling Label text changes (warnings, dosing updates)
- SUPPL - Manufacturing Production changes (new facility)
- SUPPL - Chemistry Formulation changes (new dosage strength)

Green lines in the timeline show ORIG and Efficacy approvals - the clinically meaningful milestones.

VALTREX FDA Label Details

Indications & Usage

FDA Label (PDF)

VALTREX is a deoxynucleoside analogue DNA polymerase inhibitor indicated for: Adult Patients Cold Sores (Herpes Labialis) Genital Herpes Treatment in immunocompetent patients (initial or recurrent episode) Suppression in immunocompetent or HIV-1−infected patients Reduction of transmission Herpes Zoster Pediatric Patients Cold Sores (Herpes Labialis) Chickenpox Limitations of Use The efficacy and safety of VALTREX have not been established in immunocompromised patients other than for the suppression of genital herpes in HIV-1−infected patients. 1.1 Adult Patients Cold Sores (Herpes Labialis) VA...

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Data Sources

Data sourced from official FDA and NIH databases. Click links to verify on original sources.