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IL-1beta Inhibitors & Biosimilars

2 drugs
Immunology
Target Attractiveness: Attractive (75%)

About IL-1beta

Interleukin-1beta (IL-1beta) is a potent pro-inflammatory cytokine that plays a critical role in the body's immune response. As a signaling protein, it mediates inflammation and has become an important drug target.

Strategic Insights

ℹ️ How we calculate
  • White space opportunity in Recurrent Diffuse Large B-Cell Lymphoma with only 2 trials.
  • Emerging modalities (Fusion protein) signal innovation opportunity.
  • phase4 represents biological uncertainty with 50% completion.
Risk Signals: ℹ️
White Space Available
2
Approved Drugs
2
Companies
7
Indications
1
Therapeutic Areas
Broadest Approval
ARCALYST
KINIKSA PHARMACEUTICALS (UK), LTD.
5
approved indications

Top IL-1beta Drugs

ARCALYST
KINIKSA PHARMACEUTICALS (UK), LTD.
5 indications · 2008
KINERET
BIOVITRUM AB
4 indications · 2001
🏢

BIOVITRUM AB and KINIKSA PHARMACEUTICALS are the only two companies with approved IL-1beta drugs.

IL-1beta Drug Modality Landscape

Modalities

Biologic (other)
1
50%
Fusion protein
1
50%

Routes of Administration

💉 Injection
1
50%
💧 Other
1
50%
💡

IL-1beta requires biologic approaches (biologic (other)), likely due to its structure or location.

Small molecule IL-1beta inhibitors represent a whitespace opportunity to expand therapeutic options.

Biologics only

📈 Modality Evolution

2001 Biologic (other) (KINERET)
2008 Fusion protein (ARCALYST)

other biologics pioneered IL-1beta targeting (2001), with fusion proteins entering more recently (2008).

2 drugs pre-2015

IL-1beta Clinical Trials 146 trials

146
Total Trials
31
Active
86
Completed
75%
Completion Rate

Completion by Phase

Phase Total Completed Failed Active Completion
Phase 1 37 22 9 6 71%
Phase 2 77 49 13 14 79%
Phase 3 25 13 4 8 76%
Phase 4 7 2 2 3 50%

Top Sponsors

Virginia Commonwealth Univer... 15 77%
Assistance Publique - Hôpita... 10 100%
Hellenic Institute for the S... 7 100%
University Hospital, Basel, ... 6 67%
Swedish Orphan Biovitrum 5 33%
Regeneron Pharmaceuticals 5 80%
Radboud University Medical C... 4 100%
University of North Carolina... 4 0%

By Modality

Small molecule
129 72%
Fusion protein
17 94%
Source: ClinicalTrials.gov · Completion rate = completed ÷ (completed + terminated + withdrawn)

Pro Intelligence Preview

Deep insights for drug target analysis

Competitive Landscape

  • 2 companies competing
  • Market share by company

Full Drug Portfolio

  • All 2 approved drugs
  • Approval dates & indications

Genetic Validation

  • Full genetic evidence table
  • Effect sizes & directions

Approval Timeline

  • Full 2-drug timeline
  • First-of-modality markers

Clinical Trials Analysis

  • Competition: High (15 sponsors)
  • White space: 10 underexplored indications
  • Success rates by condition
Unlock Full Intelligence

Full summary • All drugs • Genetic evidence • Trials • Timeline

How We Calculate These Metrics

Target Attractiveness Score

A 0-100 score based on trial activity, sponsor diversity, and completion rates. Calculated from 107 clinical trials targeting IL-1beta.

Completion rate: Percentage of trials that reached their planned endpoint. Trials terminated early, withdrawn, or suspended are not counted—these often indicate safety issues, lack of efficacy, or strategic pivots.

  • Highly Attractive (80+): High trial activity, many sponsors, strong completion rates
  • Attractive (60-79): Good trial activity and validation
  • Moderate (40-59): Moderate interest from sponsors
  • Low (under 40): Limited trial activity or validation concerns

Strategic Insights

Auto-generated insights based on trial analytics including competition intensity, white space opportunities, modality shifts, and failure patterns. We analyze trial sponsors, phases, indications, and outcomes.

Risk Signals

  • High Competition: Many sponsors competing for this target (may reduce market opportunity)
  • High Failure Risk: Low trial completion rates suggest development challenges
  • Low Validation: Limited trial activity or poor outcomes indicate uncertain viability
  • White Space Available: Underexplored indications present opportunities